平安! 发表于 2011-11-9 19:57 ) U' ~0 X; z+ }7 G: ?
Pazopanib (100 mg/kg/day free base equivalent) ! f* X9 d( M$ Q/ f
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。( X& U; K2 |. Q; ^' z
搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。& h4 K. C* U. n" l( Z) k7 |, w
6 n4 B3 |# Q0 m; w+ i+ V$ \以下是正版说明书的推荐用量。
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7 p' t+ Q$ P7 K+ h; p. P0 _--------------------- DOSAGE AND ADMINISTRATION ----------------# @ E5 C- _& }! k2 a$ V# i
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
9 [; l, L# o n$ n( Z* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) % x J% b8 w4 ?; W/ B) r
---------------------DOSAGE FORMS AND STRENGTHS --------------* @* r; T7 ?3 A$ i5 F$ L# C
200 mg tablets. (3) & @/ f/ G( ` o! F6 r0 b
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