平安! 发表于 2011-11-9 19:57
' b1 F8 [/ p) J* g5 _& yPazopanib (100 mg/kg/day free base equivalent)
8 w. J% @5 p- S( B+ ? 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。3 h7 K1 \( G5 a
搜索了一下,原料一大堆。
7 k8 V3 L. J/ h( q) l6 V
1 T6 x! M6 D( X& ~" q: x2 w. w对不起!100mg/kg是用于移植瘤的,我弄错了。+ C$ k9 g: J' N# X9 C
5 K6 Y$ q! Z; v D+ V8 i以下是正版说明书的推荐用量。5 n" T% E* d& o, k5 P. i" }
. T% a( w0 t: B( {" T% U7 D) I) P) o0 t
--------------------- DOSAGE AND ADMINISTRATION ----------------
f0 `" m& _/ u" V* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
/ A& r/ N, H9 v. [* M6 u6 G W/ U* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) * r) T! Q! h' b7 ]) V% |$ f( `# U1 z
---------------------DOSAGE FORMS AND STRENGTHS --------------& s/ Q" I& Z) q. W
200 mg tablets. (3) ' o: b7 _3 j# ~$ P: W
-------------------------------CONTRAINDICATIONS------------------------ |