平安! 发表于 2011-11-9 19:57
9 p) a" w3 u4 Y7 U( l# ~4 DPazopanib (100 mg/kg/day free base equivalent)
- G8 ?' d% D: N8 r _# g 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。2 x2 M' T7 B' F5 D; M! z- m
搜索了一下,原料一大堆。
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5 |( q3 X9 N$ S2 r/ v" C: d! j$ |( X对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。( u! N* R1 ?: u6 ?
3 v% e" Z# G- }) t+ ?6 P5 A' e--------------------- DOSAGE AND ADMINISTRATION ----------------
8 t; ? j0 s c2 m* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
: v& O# ?/ G* Q6 G* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) 0 m" f) W/ P1 C5 |( X1 G# j9 d' U
---------------------DOSAGE FORMS AND STRENGTHS --------------) u/ E, g/ C* L9 L: w6 |
200 mg tablets. (3) ^8 \( n3 v! k9 P1 \, z0 i3 u
-------------------------------CONTRAINDICATIONS------------------------ |