平安! 发表于 2011-11-9 19:57
9 L; p8 M6 j3 |# N. ZPazopanib (100 mg/kg/day free base equivalent)
3 x% k. _3 h6 W- M 这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
4 g6 O2 S* C; m搜索了一下,原料一大堆。
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$ R! M; ~. K2 y5 U对不起!100mg/kg是用于移植瘤的,我弄错了。
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' z: ?! N+ }+ q. ]5 A1 P& j以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------5 \* S5 _. k' E! d
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) , Z2 p& h9 [8 |8 f
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
# \2 S6 F9 ]5 |+ C: i---------------------DOSAGE FORMS AND STRENGTHS --------------7 R+ q: e+ ?- u0 N% V: M
200 mg tablets. (3)
5 e1 x$ {0 ]5 d* ~-------------------------------CONTRAINDICATIONS------------------------ |